Genistein - a neuroprotective treatment for brain injury arising from excessive glutamate release such as occurs with stroke and epilepsy.

Background

Traumatic brain injury is a major medical problem globally and is one of the leading causes of death and disability. There is no known treatment for stroke or ischaemic brain injury.

A stroke is a medical emergency and can cause permanent brain damage and death. Risk factors for stroke include old age, high blood pressure, previous stroke or transient ischemic attack (TIA), diabetes, high cholesterol, smoking and heart attack. Stroke is the second leading cause of death worldwide.

The Technology

This invention has arisen from our discovery of a novel isoform of the TRPC3 ion channel subunit (TRPC3c) which has notably stronger activation and associated Ca2+ entry than previously identified isoforms.  We have shown that expression of this TRPC3c isoform is regulated in the brain, and that the channel activity of TRPC3c channels is potently blocked by genistein and PyR3, another TRPC channel blocker.

Key Benefits

Currently no known treatments for stroke
TRPC3(c) drug target for ischaemic/excitotoxic brain injury
Treatment of epileptic seizures
Traumatic brain injury neuroprotection

UNSW is seeking a commercial partner to licence and/or to work collaboratively with the inventor Professor Gary Housley in the development of this potentially disruptive therapeutic agent.
 

https://research.unsw.edu.au/people/professor-gary-david-housley

 

Please click here to view a one-page Technology Brief

Patent Information:
For Information, Contact:
Joe Brennan
Business Development Manager
University of New South Wales
j.brennan@nsinnovations.com.au
Reference ID: 12_2712
Inventors:
Gary Housley
Youngsoo Kim
Paul Bertrand
Andrew Moorhouse
Ann Chi Yan Wong
Amanda Craig
John Power
Matthias Klugmann
Arun Krishnan
Renee Morris
Keywords:
Biotech
Chemical
Drug Development
Life Sciences
Medical/Clinical
Natural therapies
Pharmaceutical
Veterinarian
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